合研生物擁有豐富的酶學篩選經驗,根據樣本量的大小提供靈活的項目實施安排計劃,可提供96孔和384孔兩種板型的篩選模式,加速您的藥物研發進程。
Cat# |
Target |
Assay |
Format |
Deacetylases |
|||
E001 |
HDAC |
Fluorogenic assay |
96 well |
E002 |
HDAC1 |
Fluorogenic assay |
96 well |
E003 |
HDAC2 |
Fluorogenic assay |
96 well |
E004 |
HDAC3 |
Fluorogenic assay |
96 well |
E005 |
HDAC4 |
Fluorogenic assay |
96 well |
E006 |
HDAC5 |
Fluorogenic assay |
96 well |
E007 |
HDAC6 |
Fluorogenic assay |
96 well |
E008 |
HDAC7 |
Fluorogenic assay |
96 well |
E009 |
HDAC8 |
Fluorogenic assay |
96 well |
E010 |
HDAC9 |
Fluorogenic assay |
96 well |
E011 |
SIRT1 |
Fluorogenic assay |
96 well |
E012 |
SIRT2 |
Fluorogenic assay |
96 well |
E013 |
SIRT3 |
Fluorogenic assay |
96 well |
E014 |
SIRT5 |
Fluorogenic assay |
96 well |
Demethylases |
|||
E015 |
FBXL10 |
AlphaScreen assay/Chemiluminescent |
96/384 well |
E016 |
FBXL11 |
AlphaScreen assay |
96/384 well |
E017 |
JARID1A |
AlphaScreen assay/Chemiluminescent |
96/384 well |
E018 |
JARID1B |
AlphaScreen assay/Chemiluminescent |
96/384 well |
E019 |
JARID1C |
AlphaScreen assay |
96/384 well |
E020 |
JHDM1D |
AlphaScreen assay/Chemiluminescent |
96/384 well |
E021 |
JMJD1A |
AlphaScreen assay |
96/384 well |
E022 |
LSD1 |
Fluorogenic assay |
96/384 well |
E023 |
JMJD2A |
AlphaScreen assay |
96/384 well |
E024 |
JMJD2B |
AlphaScreen assay |
96/384 well |
E025 |
JMJD2C |
AlphaScreen assay/Chemiluminescent |
96/384 well |
E026 |
JMJD2D |
Chemiluminescent assay |
96/384 well |
E027 |
JMJD2E |
AlphaScreen assay |
96/384 well |
E028 |
JMJD3 |
AlphaScreen assay/Chemiluminescent |
96/384 well |
E029 |
PHF8 |
AlphaScreen assay |
96/384 well |
E030 |
TET1 |
Chemiluminescent assay |
96 well |
E031 |
TET2 |
Chemiluminescent assay |
96 well |
E032 |
UTX |
AlphaScreen assay/Chemiluminescent |
96/384 well |
Methyltransferases |
|||
E033 |
DNMT |
chemiluminescence |
96 well |
E034 |
DNMT1 |
chemiluminescence |
96 well |
E035 |
DNMT3A |
chemiluminescence |
96 well |
E036 |
DNMT3B |
chemiluminescence |
96 well |
E037 |
DOT1L |
chemiluminescence |
96 well |
E038 |
EHMT1/GLP |
chemiluminescence |
96 well |
E039 |
EZH1 |
chemiluminescence |
96 well |
E040 |
EZH2(A677G) |
chemiluminescence |
96 well |
E041 |
EZH2(Y641F) |
chemiluminescence |
96 well |
E042 |
EZH2(A641N) |
chemiluminescence/TR-FRET |
96 well |
E043 |
G9a |
chemiluminescence |
96 well |
E044 |
Histone H3(K9) |
chemiluminescence |
96 well |
E045 |
Histone H4(R3) |
AlphaScreen assay |
96 well |
E046 |
MLL1 |
chemiluminescence |
96 well |
E047 |
NSD1 |
chemiluminescence |
96 well |
E048 |
NSD2 |
chemiluminescence |
96 well |
E049 |
PRMT1 |
chemiluminescence/AlphaScreen assay |
96 well |
E050 |
PRMT3 |
chemiluminescence/AlphaScreen assay |
96 well |
E051 |
PRMT4 |
chemiluminescence |
96 well |
E052 |
PRMT5 |
chemiluminescence/TR-FRET |
96/384 well |
E053 |
PRMT8 |
chemiluminescence |
96 well |
E054 |
SETD2 |
chemiluminescence |
96 well |
E055 |
SetDB1 |
chemiluminescence |
96 well |
E056 |
SUV39H1 |
chemiluminescence |
96 well |
E057 |
SUV39H2 |
chemiluminescence |
96 well |
E058 |
SUV4-20H1 |
chemiluminescence |
96 well |
E059 |
EZH2(A378T) |
chemiluminescence |
96 well |
E060 |
NSD3 |
chemiluminescence |
96 well |
E061 |
PRMT6 |
chemiluminescence/TR-FRET |
96/384 well |
E062 |
PRMT9 |
AlphaScreen assay |
96 well |
E063 |
SMYD2 |
chemiluminescence |
96 well |
E064 |
SMYD3 |
AlphaScreen assay |
96 well |
E065 |
SMYD4 |
chemiluminescence |
96 well |
E066 |
SET7/9 |
Fluorogenic assay |
96 well |
E067 |
SET8 |
Fluorogenic assay |
96 well |
Phosphodiesterase |
|||
E068 |
PDE |
FP Assay |
96 well |
E069 |
PDE10A |
TR-FRET |
96 well |
E070 |
PDE10A1 |
TR-FRET/ FP Assay |
96 /384 well |
E071 |
PDE10A2 |
FP Assay |
96 well |
E072 |
PDE11A |
FP Assay |
96 well |
E073 |
PDE1A |
FP Assay |
96 well |
E074 |
PDE1B |
TR-FRET |
96 well |
E075 |
PDE1C |
TR-FRET/ FP Assay |
96 /384 well |
E076 |
PDE2A |
FP Assay/ FP Assay |
96 /384 well |
E077 |
PDE3A |
TR-FRET |
96 well |
E078 |
PDE3B |
FP Assay/ FP Assay |
96 /384 well |
E079 |
PDE4A |
FP Assay |
96 well |
E080 |
PDE4B2 |
FP Assay |
96 well |
E081 |
PDE4D2 |
TR-FRET |
96 well |
E082 |
PDE4D3 |
TR-FRET |
96 well |
E083 |
PDE4D7 |
TR-FRET |
96 well |
E084 |
PDE5A1 |
FP Assay/ FP Assay |
96 /384 well |
E085 |
PDE7A |
FP Assay/ FP Assay |
96 /384 well |
E086 |
PDE7B |
FP Assay |
96 well |
E087 |
PDE8A |
FP Assay |
96 well |
E088 |
PDE9A |
FP Assay |
96 well |
E089 |
PDE4C |
FP Assay |
384 well |
E090 |
Autotaxin |
Fluorogenic assay |
96 well |
PARPs |
|||
E091 |
PARP1 |
chemiluminescence/Colorimetric Assay |
96/384 well |
E092 |
PARP2 |
chemiluminescence/Colorimetric Assay |
96/384 well |
E093 |
PARP3 |
chemiluminescence |
96/384 well |
E094 |
PARP6 |
chemiluminescence |
96/384 well |
E095 |
PARP7 |
chemiluminescence |
96/384 well |
E096 |
PARP10 |
chemiluminescence |
96/384 well |
E097 |
PARP11 |
chemiluminescence |
96/384 well |
E098 |
PARP14 |
chemiluminescence |
96/384 well |
E099 |
PARP15 |
chemiluminescence |
96/384 well |
E100 |
TNKS1 |
chemiluminescence |
96/384 well |
E101 |
TNKS2 |
chemiluminescence |
96/384 well |
Protease |
|||
E102 |
DPP3 |
Fluorogenic assay |
96 well |
E103 |
DPP4 |
Fluorogenic assay |
96 well |
E104 |
DPP7 |
Fluorogenic assay |
96 well |
E105 |
DPP8 |
Fluorogenic assay |
96 well |
E106 |
DPP9 |
Fluorogenic assay |
96 well |
E107 |
FAP |
Fluorogenic assay |
96 well |
E108 |
POP |
Fluorogenic assay |
96 well |
E109 |
Renin |
Fluorogenic assay |
96 well |
E110 |
Caspase-3 |
Fluorogenic assay |
96 well |
E111 |
Caspase-6 |
Fluorogenic assay |
96 well |
E112 |
Caspase-7 |
Fluorogenic assay |
96 well |
E113 |
Caspase-8 |
Fluorogenic assay |
96 well |
Bromodomains |
|||
E114 |
ATAD2A |
TR-FRET/AlphaScreen assay |
96/384 well |
E115 |
ATAD2B |
TR-FRET/AlphaScreen assay |
96/384 well |
E116 |
BAZ2B |
AlphaScreen assay |
96/384 well |
E117 |
BPTF/FALZ |
TR-FRET |
96/384 well |
E118 |
BRD1 |
TR-FRET/AlphaScreen assay |
96/384 well |
E119 |
BRD2 |
TR-FRET/AlphaScreen assay |
96/384 well |
E120 |
BRD3 |
TR-FRET/AlphaScreen assay |
96/384 well |
E121 |
BRD4 |
TR-FRET/AlphaScreen assay |
96/384 well |
E122 |
BRD9 |
TR-FRET |
96/384 well |
E123 |
BRDT |
TR-FRET |
96/384 well |
E124 |
BRPF3 |
TR-FRET/AlphaScreen assay |
96/384 well |
E125 |
CECR2 |
TR-FRET/AlphaScreen assay |
96/384 well |
E126 |
CREBBP |
TR-FRET/AlphaScreen assay |
96/384 well |
E127 |
SMARCA2 |
TR-FRET/AlphaScreen assay |
96/384 well |
E128 |
SMARCA4 |
TR-FRET/AlphaScreen assay |
96/384 well |
E129 |
TAF1(BD2) |
TR-FRET |
96/384 well |
E130 |
TAF1L(BD2) |
TR-FRET |
96/384 well |
E131 |
TRIM24 |
TR-FRET |
96/384 well |
E132 |
WDR9/BRWD1 |
TR-FRET |
96/384 well |
E133 |
BACE1 |
TR-FRET |
96/384 well |
E134 |
BRG1 |
TR-FRET |
96 well |
E135 |
BRM |
TR-FRET |
96 well |
E136 |
CBP |
TR-FRET |
96 well |
Kinase |
|||
E137 |
ABL1 |
ADP-Glo |
96/384 well |
E138 |
ABL1(E255K) |
ADP-Glo |
96/384 well |
E139 |
ABL1(T315I) |
ADP-Glo |
96/384 well |
E140 |
ABL1(Y253F) |
ADP-Glo |
96/384 well |
E141 |
ACK |
ADP-Glo |
96/384 well |
E142 |
AKT1 |
ADP-Glo |
96/384 well |
E143 |
AKT2 |
ADP-Glo |
96/384 well |
E144 |
AKT3 |
ADP-Glo |
96/384 well |
E145 |
ALK2 |
ADP-Glo |
96/384 well |
E146 |
ALK4 |
ADP-Glo |
96/384 well |
E147 |
ALK6 |
ADP-Glo |
96/384 well |
E148 |
AMAPK(A1/B1/G2) |
ADP-Glo |
96/384 well |
E149 |
AMPK(A1/B1/G1) |
ADP-Glo |
96/384 well |
E150 |
AMPK(A2/B1/G1) |
ADP-Glo |
96/384 well |
E151 |
ASK1 |
ADP-Glo |
96/384 well |
E152 |
Aurora A |
ADP-Glo |
96/384 well |
E153 |
Aurora B |
ADP-Glo |
96/384 well |
E154 |
AXL |
ADP-Glo |
96/384 well |
E155 |
BRK |
ADP-Glo |
96/384 well |
E156 |
BXM |
ADP-Glo |
96/384 well |
E157 |
CAMK1γ |
ADP-Glo |
96/384 well |
E158 |
CAMK2α |
ADP-Glo |
96/384 well |
E159 |
CAMK2γ |
ADP-Glo |
96/384 well |
E160 |
CAMKK1 |
ADP-Glo |
96/384 well |
E161 |
CDC7/DBF4 |
ADP-Glo |
96/384 well |
E162 |
CDK2/CyclinA2 |
ADP-Glo |
96/384 well |
E163 |
CDK2/CyclinE1 |
ADP-Glo |
96/384 well |
E164 |
CDK3/cyclinE1 |
ADP-Glo |
96/384 well |
E165 |
CDK5/p25 |
ADP-Glo |
96/384 well |
E166 |
CDK5/p35 |
ADP-Glo |
96/384 well |
E167 |
CDK6/CyclinD3 |
ADP-Glo |
96/384 well |
E168 |
CDK9/Cyclink |
ADP-Glo |
96/384 well |
E169 |
CHK1 |
ADP-Glo |
96/384 well |
E170 |
CHK2 |
ADP-Glo |
96/384 well |
E171 |
CK1a1 |
ADP-Glo |
96/384 well |
E172 |
CK1γ1 |
ADP-Glo |
96/384 well |
E173 |
CK1ε |
ADP-Glo |
96/384 well |
E174 |
CK2α1 |
ADP-Glo |
96/384 well |
E175 |
c-KIT |
ADP-Glo |
96/384 well |
E176 |
CLK1 |
ADP-Glo |
96/384 well |
E177 |
CLK3 |
ADP-Glo |
96/384 well |
E178 |
c-MER |
ADP-Glo |
96/384 well |
E179 |
CSK |
ADP-Glo |
96/384 well |
E180 |
DAPK1 |
ADP-Glo |
96/384 well |
E181 |
DDR2 |
ADP-Glo |
96/384 well |
E182 |
DNA-PK |
ADP-Glo |
96/384 well |
E183 |
DYRK2 |
ADP-Glo |
96/384 well |
E184 |
EGFR |
ADP-Glo |
96/384 well |
E185 |
EGFR(L858R) |
ADP-Glo |
96/384 well |
E186 |
EGFR(L861Q) |
ADP-Glo |
96/384 well |
E187 |
EGFR(T790,L858R) |
ADP-Glo |
96/384 well |
E188 |
EGFR(T790M) |
ADP-Glo |
96/384 well |
E189 |
EIF2AK2 |
ADP-Glo |
96/384 well |
E190 |
EPHA1 |
ADP-Glo |
96/384 well |
E191 |
ERK1 |
ADP-Glo |
96/384 well |
E192 |
ERK2 |
ADP-Glo |
96/384 well |
E193 |
FAK |
ADP-Glo |
96/384 well |
E194 |
FES |
ADP-Glo |
96/384 well |
E195 |
FGFR1 |
ADP-Glo |
96/384 well |
E196 |
FGFR2 |
ADP-Glo |
96/384 well |
E197 |
FGFR3(K650E) |
ADP-Glo |
96/384 well |
E198 |
FGFR4 |
ADP-Glo |
96/384 well |
E199 |
FLT1 |
ADP-Glo |
96/384 well |
E200 |
FLT3 |
ADP-Glo |
96/384 well |
E201 |
FLT3(D835Y) |
ADP-Glo |
96/384 well |
E202 |
FMS |
ADP-Glo |
96/384 well |
E203 |
FYN A |
ADP-Glo |
96/384 well |
E204 |
GRK5 |
ADP-Glo |
96/384 well |
E205 |
GSK3α |
ADP-Glo |
96/384 well |
E206 |
GSK3β |
ADP-Glo |
96/384 well |
E207 |
HER2 |
ADP-Glo |
96/384 well |
E208 |
HER4 |
ADP-Glo |
96/384 well |
E209 |
HIPK1 |
ADP-Glo |
96/384 well |
E210 |
HPK1 |
ADP-Glo |
96/384 well |
E211 |
IGF1R |
ADP-Glo |
96/384 well |
E212 |
IKK |
ADP-Glo |
96/384 well |
E213 |
IKKα |
ADP-Glo |
96/384 well |
E214 |
InsR |
ADP-Glo |
96/384 well |
E215 |
IRAK4 |
ADP-Glo |
96/384 well |
E216 |
ITK |
ADP-Glo |
96/384 well |
E217 |
JAK3 |
ADP-Glo |
96/384 well |
E218 |
JNK1 |
ADP-Glo |
96/384 well |
E219 |
JNK3 |
ADP-Glo |
96/384 well |
E220 |
KDR |
ADP-Glo |
96/384 well |
E221 |
KHS1 |
ADP-Glo |
96/384 well |
E222 |
LCK |
ADP-Glo |
96/384 well |
E223 |
Lipid kinase |
ADP-Glo |
96/384 well |
E224 |
LRRK2 |
ADP-Glo |
96/384 well |
E225 |
LYN B |
ADP-Glo |
96/384 well |
E226 |
MAPKAPK2 |
ADP-Glo |
96/384 well |
E227 |
MAPKAPK3 |
ADP-Glo |
96/384 well |
E228 |
MAPKAPK5 |
ADP-Glo |
96/384 well |
E229 |
MARK1 |
ADP-Glo |
96/384 well |
E230 |
MELK |
ADP-Glo |
96/384 well |
E231 |
MET |
ADP-Glo |
96/384 well |
E232 |
MET(M1250T) |
ADP-Glo |
96/384 well |
E233 |
MINK1 |
ADP-Glo |
96/384 well |
E234 |
MLCK |
ADP-Glo |
96/384 well |
E235 |
MLK1 |
ADP-Glo |
96/384 well |
E236 |
MLK2 |
ADP-Glo |
96/384 well |
E237 |
MRCKa |
ADP-Glo |
96/384 well |
E238 |
MSK1 |
ADP-Glo |
96/384 well |
E239 |
MSK2 |
ADP-Glo |
96/384 well |
E240 |
MST1 |
ADP-Glo |
96/384 well |
E241 |
MYO3β |
ADP-Glo |
96/384 well |
E242 |
Name |
ADP-Glo |
96/384 well |
E243 |
NEK2 |
ADP-Glo |
96/384 well |
E244 |
NEK3 |
ADP-Glo |
96/384 well |
E245 |
NIK |
ADP-Glo |
96/384 well |
E246 |
NUAK2 |
ADP-Glo |
96/384 well |
E247 |
p38α |
ADP-Glo |
96/384 well |
E248 |
p38B |
ADP-Glo |
96/384 well |
E249 |
p38γ |
ADP-Glo |
96/384 well |
E250 |
P38δ |
ADP-Glo |
96/384 well |
E251 |
p70S6K |
ADP-Glo |
96/384 well |
E252 |
p70S6Kb |
ADP-Glo |
96/384 well |
E253 |
PAK1/CDC42 |
ADP-Glo |
96/384 well |
E254 |
PAK3 |
ADP-Glo |
96/384 well |
E255 |
PAK4 |
ADP-Glo |
96/384 well |
E256 |
PASK |
ADP-Glo |
96/384 well |
E257 |
PDGFRa(D842V) |
ADP-Glo |
96/384 well |
E258 |
PDGFRa(T674I) |
ADP-Glo |
96/384 well |
E259 |
PDGFRα |
ADP-Glo |
96/384 well |
E260 |
PDGFRβ |
ADP-Glo |
96/384 well |
E261 |
PDK1 |
ADP-Glo |
96/384 well |
E262 |
PI3K Lipid kinases |
ADP-Glo |
96/384 well |
E263 |
PI3K-Glo |
ADP-Glo |
96/384 well |
E264 |
PIM1 |
ADP-Glo |
96/384 well |
E265 |
PIM2 |
ADP-Glo |
96/384 well |
E266 |
PKA |
ADP-Glo |
96/384 well |
E267 |
PKC |
ADP-Glo |
96/384 well |
E268 |
PKC1 |
ADP-Glo |
96/384 well |
E269 |
PKCα |
ADP-Glo |
96/384 well |
E270 |
PKCβII |
ADP-Glo |
96/384 well |
E271 |
PKCγ |
ADP-Glo |
96/384 well |
E272 |
PKCδ |
ADP-Glo |
96/384 well |
E273 |
PKCε |
ADP-Glo |
96/384 well |
E274 |
PKCζ |
ADP-Glo |
96/384 well |
E275 |
PKCθ |
ADP-Glo |
96/384 well |
E276 |
PKCι |
ADP-Glo |
96/384 well |
E277 |
PKCμ |
ADP-Glo |
96/384 well |
E278 |
PKD2 |
ADP-Glo |
96/384 well |
E279 |
PLK1 |
ADP-Glo |
96/384 well |
E280 |
PRKG1 |
ADP-Glo |
96/384 well |
E281 |
PYK2 |
ADP-Glo |
96/384 well |
E282 |
RET |
ADP-Glo |
96/384 well |
E283 |
RET(V804L) |
ADP-Glo |
96/384 well |
E284 |
RET(Y791F) |
ADP-Glo |
96/384 well |
E285 |
RIPK2 |
ADP-Glo |
96/384 well |
E286 |
ROCK1 |
ADP-Glo |
96/384 well |
E287 |
ROCK2 |
ADP-Glo |
96/384 well |
E288 |
RON |
ADP-Glo |
96/384 well |
E289 |
RSK1 |
ADP-Glo |
96/384 well |
E290 |
SGK1 |
ADP-Glo |
96/384 well |
E291 |
SIK |
ADP-Glo |
96/384 well |
E292 |
SLK |
ADP-Glo |
96/384 well |
E293 |
SRC |
ADP-Glo |
96/384 well |
E294 |
STK33 |
ADP-Glo |
96/384 well |
E295 |
SYK |
ADP-Glo |
96/384 well |
E296 |
TAK1-TAB1 |
ADP-Glo |
96/384 well |
E297 |
TAOK1 |
ADP-Glo |
96/384 well |
E298 |
TBK1 |
ADP-Glo |
96/384 well |
E299 |
TGFbR1 |
ADP-Glo |
96/384 well |
E300 |
TGFβR2 |
ADP-Glo |
96/384 well |
E301 |