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    酶學靶點篩選

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    所在地: 湖北武漢市
    有效期至: 長期有效
    最后更新: 2018-08-20 13:40
    瀏覽次數: 488
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    服務說明
     分子靶點篩選的藥物發現途徑越來越廣泛的運用于新藥的開發中,酶學研究在新藥研發中的地位越來越重要。酶學實驗涵蓋600多種篩選模型,包括了常見的組蛋白去乙酰酶類,組蛋白去甲基化酶,酪氨酸激酶,絲氨酸激酶,甲基化轉移酶,磷酸二酯酶,DNA修復酶,熱休克蛋白,免疫相關蛋白等,以及激酶譜的篩選。
    合研生物擁有豐富的酶學篩選經驗,根據樣本量的大小提供靈活的項目實施安排計劃,可提供96孔和384孔兩種板型的篩選模式,加速您的藥物研發進程。

     

    Cat#

    Target

    Assay

    Format

    Deacetylases

    E001

    HDAC

    Fluorogenic assay

    96 well

    E002

    HDAC1

    Fluorogenic assay

    96 well

    E003

    HDAC2

    Fluorogenic assay

    96 well

    E004

    HDAC3

    Fluorogenic assay

    96 well

    E005

    HDAC4

    Fluorogenic assay

    96 well

    E006

    HDAC5

    Fluorogenic assay

    96 well

    E007

    HDAC6

    Fluorogenic assay

    96 well

    E008

    HDAC7

    Fluorogenic assay

    96 well

    E009

    HDAC8

    Fluorogenic assay

    96 well

    E010

    HDAC9

    Fluorogenic assay

    96 well

    E011

    SIRT1

    Fluorogenic assay

    96 well

    E012

    SIRT2

    Fluorogenic assay

    96 well

    E013

    SIRT3

    Fluorogenic assay

    96 well

    E014

    SIRT5

    Fluorogenic assay

    96 well

    Demethylases

    E015

    FBXL10

    AlphaScreen assay/Chemiluminescent

    96/384 well

    E016

    FBXL11

    AlphaScreen assay

    96/384 well

    E017

    JARID1A

    AlphaScreen assay/Chemiluminescent

    96/384 well

    E018

    JARID1B

    AlphaScreen assay/Chemiluminescent

    96/384 well

    E019

    JARID1C

    AlphaScreen assay

    96/384 well

    E020

    JHDM1D

    AlphaScreen assay/Chemiluminescent

    96/384 well

    E021

    JMJD1A

    AlphaScreen assay

    96/384 well

    E022

    LSD1

    Fluorogenic assay

    96/384 well

    E023

    JMJD2A

    AlphaScreen assay

    96/384 well

    E024

    JMJD2B

    AlphaScreen assay

    96/384 well

    E025

    JMJD2C

    AlphaScreen assay/Chemiluminescent

    96/384 well

    E026

    JMJD2D

    Chemiluminescent assay

    96/384 well

    E027

    JMJD2E

    AlphaScreen assay

    96/384 well

    E028

    JMJD3

    AlphaScreen assay/Chemiluminescent

    96/384 well

    E029

    PHF8

    AlphaScreen assay

    96/384 well

    E030

    TET1

    Chemiluminescent assay

    96 well

    E031

    TET2

    Chemiluminescent assay

    96 well

    E032

    UTX

    AlphaScreen assay/Chemiluminescent

    96/384 well

    Methyltransferases

    E033

    DNMT

    chemiluminescence

    96 well

    E034

    DNMT1

    chemiluminescence

    96 well

    E035

    DNMT3A

    chemiluminescence

    96 well

    E036

    DNMT3B

    chemiluminescence

    96 well

    E037

    DOT1L

    chemiluminescence

    96 well

    E038

    EHMT1/GLP

    chemiluminescence

    96 well

    E039

    EZH1

    chemiluminescence

    96 well

    E040

    EZH2(A677G)

    chemiluminescence

    96 well

    E041

    EZH2(Y641F)

    chemiluminescence

    96 well

    E042

    EZH2(A641N)

    chemiluminescence/TR-FRET

    96 well

    E043

    G9a

    chemiluminescence

    96 well

    E044

    Histone H3(K9)

    chemiluminescence

    96 well

    E045

    Histone H4(R3)

    AlphaScreen assay

    96 well

    E046

    MLL1

    chemiluminescence

    96 well

    E047

    NSD1

    chemiluminescence

    96 well

    E048

    NSD2

    chemiluminescence

    96 well

    E049

    PRMT1

    chemiluminescence/AlphaScreen assay

    96 well

    E050

    PRMT3

    chemiluminescence/AlphaScreen assay

    96 well

    E051

    PRMT4

    chemiluminescence

    96 well

    E052

    PRMT5

    chemiluminescence/TR-FRET

    96/384 well

    E053

    PRMT8

    chemiluminescence

    96 well

    E054

    SETD2

    chemiluminescence

    96 well

    E055

    SetDB1

    chemiluminescence

    96 well

    E056

    SUV39H1

    chemiluminescence

    96 well

    E057

    SUV39H2

    chemiluminescence

    96 well

    E058

    SUV4-20H1

    chemiluminescence

    96 well

    E059

    EZH2(A378T)

    chemiluminescence

    96 well

    E060

    NSD3

    chemiluminescence

    96 well

    E061

    PRMT6

    chemiluminescence/TR-FRET

    96/384 well

    E062

    PRMT9

    AlphaScreen assay

    96 well

    E063

    SMYD2

    chemiluminescence

    96 well

    E064

    SMYD3

    AlphaScreen assay

    96 well

    E065

    SMYD4

    chemiluminescence

    96 well

    E066

    SET7/9

    Fluorogenic assay

    96 well

    E067

    SET8

    Fluorogenic assay

    96 well

    Phosphodiesterase

    E068

    PDE

    FP Assay

    96 well

    E069

    PDE10A

    TR-FRET

    96 well

    E070

    PDE10A1

    TR-FRET/ FP Assay

    96 /384 well

    E071

    PDE10A2

    FP Assay

    96 well

    E072

    PDE11A

    FP Assay

    96 well

    E073

    PDE1A

    FP Assay

    96 well

    E074

    PDE1B

    TR-FRET

    96 well

    E075

    PDE1C

    TR-FRET/ FP Assay

    96 /384 well

    E076

    PDE2A

    FP Assay/ FP Assay

    96 /384 well

    E077

    PDE3A

    TR-FRET

    96 well

    E078

    PDE3B

    FP Assay/ FP Assay

    96 /384 well

    E079

    PDE4A

    FP Assay

    96 well

    E080

    PDE4B2

    FP Assay

    96 well

    E081

    PDE4D2

    TR-FRET

    96 well

    E082

    PDE4D3

    TR-FRET

    96 well

    E083

    PDE4D7

    TR-FRET

    96 well

    E084

    PDE5A1

    FP Assay/ FP Assay

    96 /384 well

    E085

    PDE7A

    FP Assay/ FP Assay

    96 /384 well

    E086

    PDE7B

    FP Assay

    96 well

    E087

    PDE8A

    FP Assay

    96 well

    E088

    PDE9A

    FP Assay

    96 well

    E089

    PDE4C

    FP Assay

    384 well

    E090

    Autotaxin

    Fluorogenic assay

    96 well

    PARPs

    E091

    PARP1

    chemiluminescence/Colorimetric Assay

    96/384 well

    E092

    PARP2

    chemiluminescence/Colorimetric Assay

    96/384 well

    E093

    PARP3

    chemiluminescence

    96/384 well

    E094

    PARP6

    chemiluminescence

    96/384 well

    E095

    PARP7

    chemiluminescence

    96/384 well

    E096

    PARP10

    chemiluminescence

    96/384 well

    E097

    PARP11

    chemiluminescence

    96/384 well

    E098

    PARP14

    chemiluminescence

    96/384 well

    E099

    PARP15

    chemiluminescence

    96/384 well

    E100

    TNKS1

    chemiluminescence

    96/384 well

    E101

    TNKS2

    chemiluminescence

    96/384 well

    Protease

    E102

    DPP3

    Fluorogenic assay

    96 well

    E103

    DPP4

    Fluorogenic assay

    96 well

    E104

    DPP7

    Fluorogenic assay

    96 well

    E105

    DPP8

    Fluorogenic assay

    96 well

    E106

    DPP9

    Fluorogenic assay

    96 well

    E107

    FAP

    Fluorogenic assay

    96 well

    E108

    POP

    Fluorogenic assay

    96 well

    E109

    Renin

    Fluorogenic assay

    96 well

    E110

    Caspase-3

    Fluorogenic assay

    96 well

    E111

    Caspase-6

    Fluorogenic assay

    96 well

    E112

    Caspase-7

    Fluorogenic assay

    96 well

    E113

    Caspase-8

    Fluorogenic assay

    96 well

    Bromodomains

    E114

    ATAD2A

    TR-FRET/AlphaScreen assay

    96/384 well

    E115

    ATAD2B

    TR-FRET/AlphaScreen assay

    96/384 well

    E116

    BAZ2B

    AlphaScreen assay

    96/384 well

    E117

    BPTF/FALZ

    TR-FRET

    96/384 well

    E118

    BRD1

    TR-FRET/AlphaScreen assay

    96/384 well

    E119

    BRD2

    TR-FRET/AlphaScreen assay

    96/384 well

    E120

    BRD3

    TR-FRET/AlphaScreen assay

    96/384 well

    E121

    BRD4

    TR-FRET/AlphaScreen assay

    96/384 well

    E122

    BRD9

    TR-FRET

    96/384 well

    E123

    BRDT

    TR-FRET

    96/384 well

    E124

    BRPF3

    TR-FRET/AlphaScreen assay

    96/384 well

    E125

    CECR2

    TR-FRET/AlphaScreen assay

    96/384 well

    E126

    CREBBP

    TR-FRET/AlphaScreen assay

    96/384 well

    E127

    SMARCA2

    TR-FRET/AlphaScreen assay

    96/384 well

    E128

    SMARCA4

    TR-FRET/AlphaScreen assay

    96/384 well

    E129

    TAF1(BD2)

    TR-FRET

    96/384 well

    E130

    TAF1L(BD2)

    TR-FRET

    96/384 well

    E131

    TRIM24

    TR-FRET

    96/384 well

    E132

    WDR9/BRWD1

    TR-FRET

    96/384 well

    E133

    BACE1

    TR-FRET

    96/384 well

    E134

    BRG1

    TR-FRET

    96 well

    E135

    BRM

    TR-FRET

    96 well

    E136

    CBP

    TR-FRET

    96 well

    Kinase

    E137

    ABL1

    ADP-Glo

    96/384 well

    E138

    ABL1(E255K)

    ADP-Glo

    96/384 well

    E139

    ABL1(T315I)

    ADP-Glo

    96/384 well

    E140

    ABL1(Y253F)

    ADP-Glo

    96/384 well

    E141

    ACK

    ADP-Glo

    96/384 well

    E142

    AKT1

    ADP-Glo

    96/384 well

    E143

    AKT2

    ADP-Glo

    96/384 well

    E144

    AKT3

    ADP-Glo

    96/384 well

    E145

    ALK2

    ADP-Glo

    96/384 well

    E146

    ALK4

    ADP-Glo

    96/384 well

    E147

    ALK6

    ADP-Glo

    96/384 well

    E148

    AMAPK(A1/B1/G2)

    ADP-Glo

    96/384 well

    E149

    AMPK(A1/B1/G1)

    ADP-Glo

    96/384 well

    E150

    AMPK(A2/B1/G1)

    ADP-Glo

    96/384 well

    E151

    ASK1

    ADP-Glo

    96/384 well

    E152

    Aurora A

    ADP-Glo

    96/384 well

    E153

    Aurora B

    ADP-Glo

    96/384 well

    E154

    AXL

    ADP-Glo

    96/384 well

    E155

    BRK

    ADP-Glo

    96/384 well

    E156

    BXM

    ADP-Glo

    96/384 well

    E157

    CAMK1γ

    ADP-Glo

    96/384 well

    E158

    CAMK2α

    ADP-Glo

    96/384 well

    E159

    CAMK2γ

    ADP-Glo

    96/384 well

    E160

    CAMKK1

    ADP-Glo

    96/384 well

    E161

    CDC7/DBF4

    ADP-Glo

    96/384 well

    E162

    CDK2/CyclinA2

    ADP-Glo

    96/384 well

    E163

    CDK2/CyclinE1

    ADP-Glo

    96/384 well

    E164

    CDK3/cyclinE1

    ADP-Glo

    96/384 well

    E165

    CDK5/p25

    ADP-Glo

    96/384 well

    E166

    CDK5/p35

    ADP-Glo

    96/384 well

    E167

    CDK6/CyclinD3

    ADP-Glo

    96/384 well

    E168

    CDK9/Cyclink

    ADP-Glo

    96/384 well

    E169

    CHK1

    ADP-Glo

    96/384 well

    E170

    CHK2

    ADP-Glo

    96/384 well

    E171

    CK1a1

    ADP-Glo

    96/384 well

    E172

    CK1γ1

    ADP-Glo

    96/384 well

    E173

    CK1ε

    ADP-Glo

    96/384 well

    E174

    CK2α1

    ADP-Glo

    96/384 well

    E175

    c-KIT

    ADP-Glo

    96/384 well

    E176

    CLK1

    ADP-Glo

    96/384 well

    E177

    CLK3

    ADP-Glo

    96/384 well

    E178

    c-MER

    ADP-Glo

    96/384 well

    E179

    CSK

    ADP-Glo

    96/384 well

    E180

    DAPK1

    ADP-Glo

    96/384 well

    E181

    DDR2

    ADP-Glo

    96/384 well

    E182

    DNA-PK

    ADP-Glo

    96/384 well

    E183

    DYRK2

    ADP-Glo

    96/384 well

    E184

    EGFR

    ADP-Glo

    96/384 well

    E185

    EGFR(L858R)

    ADP-Glo

    96/384 well

    E186

    EGFR(L861Q)

    ADP-Glo

    96/384 well

    E187

    EGFR(T790,L858R)

    ADP-Glo

    96/384 well

    E188

    EGFR(T790M)

    ADP-Glo

    96/384 well

    E189

    EIF2AK2

    ADP-Glo

    96/384 well

    E190

    EPHA1

    ADP-Glo

    96/384 well

    E191

    ERK1

    ADP-Glo

    96/384 well

    E192

    ERK2

    ADP-Glo

    96/384 well

    E193

    FAK

    ADP-Glo

    96/384 well

    E194

    FES

    ADP-Glo

    96/384 well

    E195

    FGFR1

    ADP-Glo

    96/384 well

    E196

    FGFR2

    ADP-Glo

    96/384 well

    E197

    FGFR3(K650E)

    ADP-Glo

    96/384 well

    E198

    FGFR4

    ADP-Glo

    96/384 well

    E199

    FLT1

    ADP-Glo

    96/384 well

    E200

    FLT3

    ADP-Glo

    96/384 well

    E201

    FLT3(D835Y)

    ADP-Glo

    96/384 well

    E202

    FMS

    ADP-Glo

    96/384 well

    E203

    FYN A

    ADP-Glo

    96/384 well

    E204

    GRK5

    ADP-Glo

    96/384 well

    E205

    GSK3α

    ADP-Glo

    96/384 well

    E206

    GSK3β

    ADP-Glo

    96/384 well

    E207

    HER2

    ADP-Glo

    96/384 well

    E208

    HER4

    ADP-Glo

    96/384 well

    E209

    HIPK1

    ADP-Glo

    96/384 well

    E210

    HPK1

    ADP-Glo

    96/384 well

    E211

    IGF1R

    ADP-Glo

    96/384 well

    E212

    IKK

    ADP-Glo

    96/384 well

    E213

    IKKα

    ADP-Glo

    96/384 well

    E214

    InsR

    ADP-Glo

    96/384 well

    E215

    IRAK4

    ADP-Glo

    96/384 well

    E216

    ITK

    ADP-Glo

    96/384 well

    E217

    JAK3

    ADP-Glo

    96/384 well

    E218

    JNK1

    ADP-Glo

    96/384 well

    E219

    JNK3

    ADP-Glo

    96/384 well

    E220

    KDR

    ADP-Glo

    96/384 well

    E221

    KHS1

    ADP-Glo

    96/384 well

    E222

    LCK

    ADP-Glo

    96/384 well

    E223

    Lipid kinase

    ADP-Glo

    96/384 well

    E224

    LRRK2

    ADP-Glo

    96/384 well

    E225

    LYN B

    ADP-Glo

    96/384 well

    E226

    MAPKAPK2

    ADP-Glo

    96/384 well

    E227

    MAPKAPK3

    ADP-Glo

    96/384 well

    E228

    MAPKAPK5

    ADP-Glo

    96/384 well

    E229

    MARK1

    ADP-Glo

    96/384 well

    E230

    MELK

    ADP-Glo

    96/384 well

    E231

    MET

    ADP-Glo

    96/384 well

    E232

    MET(M1250T)

    ADP-Glo

    96/384 well

    E233

    MINK1

    ADP-Glo

    96/384 well

    E234

    MLCK

    ADP-Glo

    96/384 well

    E235

    MLK1

    ADP-Glo

    96/384 well

    E236

    MLK2

    ADP-Glo

    96/384 well

    E237

    MRCKa

    ADP-Glo

    96/384 well

    E238

    MSK1

    ADP-Glo

    96/384 well

    E239

    MSK2

    ADP-Glo

    96/384 well

    E240

    MST1

    ADP-Glo

    96/384 well

    E241

    MYO3β

    ADP-Glo

    96/384 well

    E242

    Name

    ADP-Glo

    96/384 well

    E243

    NEK2

    ADP-Glo

    96/384 well

    E244

    NEK3

    ADP-Glo

    96/384 well

    E245

    NIK

    ADP-Glo

    96/384 well

    E246

    NUAK2

    ADP-Glo

    96/384 well

    E247

    p38α

    ADP-Glo

    96/384 well

    E248

    p38B

    ADP-Glo

    96/384 well

    E249

    p38γ

    ADP-Glo

    96/384 well

    E250

    P38δ

    ADP-Glo

    96/384 well

    E251

    p70S6K

    ADP-Glo

    96/384 well

    E252

    p70S6Kb

    ADP-Glo

    96/384 well

    E253

    PAK1/CDC42

    ADP-Glo

    96/384 well

    E254

    PAK3

    ADP-Glo

    96/384 well

    E255

    PAK4

    ADP-Glo

    96/384 well

    E256

    PASK

    ADP-Glo

    96/384 well

    E257

    PDGFRa(D842V)

    ADP-Glo

    96/384 well

    E258

    PDGFRa(T674I)

    ADP-Glo

    96/384 well

    E259

    PDGFRα

    ADP-Glo

    96/384 well

    E260

    PDGFRβ

    ADP-Glo

    96/384 well

    E261

    PDK1

    ADP-Glo

    96/384 well

    E262

    PI3K Lipid kinases

    ADP-Glo

    96/384 well

    E263

    PI3K-Glo

    ADP-Glo

    96/384 well

    E264

    PIM1

    ADP-Glo

    96/384 well

    E265

    PIM2

    ADP-Glo

    96/384 well

    E266

    PKA

    ADP-Glo

    96/384 well

    E267

    PKC

    ADP-Glo

    96/384 well

    E268

    PKC1

    ADP-Glo

    96/384 well

    E269

    PKCα

    ADP-Glo

    96/384 well

    E270

    PKCβII

    ADP-Glo

    96/384 well

    E271

    PKCγ

    ADP-Glo

    96/384 well

    E272

    PKCδ

    ADP-Glo

    96/384 well

    E273

    PKCε

    ADP-Glo

    96/384 well

    E274

    PKCζ

    ADP-Glo

    96/384 well

    E275

    PKCθ

    ADP-Glo

    96/384 well

    E276

    PKCι

    ADP-Glo

    96/384 well

    E277

    PKCμ

    ADP-Glo

    96/384 well

    E278

    PKD2

    ADP-Glo

    96/384 well

    E279

    PLK1

    ADP-Glo

    96/384 well

    E280

    PRKG1

    ADP-Glo

    96/384 well

    E281

    PYK2

    ADP-Glo

    96/384 well

    E282

    RET

    ADP-Glo

    96/384 well

    E283

    RET(V804L)

    ADP-Glo

    96/384 well

    E284

    RET(Y791F)

    ADP-Glo

    96/384 well

    E285

    RIPK2

    ADP-Glo

    96/384 well

    E286

    ROCK1

    ADP-Glo

    96/384 well

    E287

    ROCK2

    ADP-Glo

    96/384 well

    E288

    RON

    ADP-Glo

    96/384 well

    E289

    RSK1

    ADP-Glo

    96/384 well

    E290

    SGK1

    ADP-Glo

    96/384 well

    E291

    SIK

    ADP-Glo

    96/384 well

    E292

    SLK

    ADP-Glo

    96/384 well

    E293

    SRC

    ADP-Glo

    96/384 well

    E294

    STK33

    ADP-Glo

    96/384 well

    E295

    SYK

    ADP-Glo

    96/384 well

    E296

    TAK1-TAB1

    ADP-Glo

    96/384 well

    E297

    TAOK1

    ADP-Glo

    96/384 well

    E298

    TBK1

    ADP-Glo

    96/384 well

    E299

    TGFbR1

    ADP-Glo

    96/384 well

    E300

    TGFβR2

    ADP-Glo

    96/384 well

    E301